Lead Optimization – Building Efficacy & Safety

May 29, 2014
Drug Discovery Series Part 4 of 8

bottle of spilled blue pills

How do you safely and effectively develop drug leads? Join Dr. Craig Lindsley, Director of the Vanderbilt Center for Neuroscience Drug Discovery as he shares strategies on how to effectively optimize small molecule hits and rapidly assess your findings in the 4th session of our Drug Discovery Series.  

What You Will Learn 

  • Strategies to efficiently optimize (med chem and DMPK) small molecule hits
  • Efficient approaches for rapid DMPK assessment and IVIVC
  • Iterative parallel synthesis and developing allosteric ligands

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The Fine Print

ACS Webinars® does not endorse any products or services. The views expressed in this presentation are those of the presenters and do not necessarily reflect the views or policies of the American Chemical Society.

ACS Webinars


Craig Lindsley
Vanderbelt Center for Neuroscience Drug Discovery